ES8700255A1 - Un procedimiento para la preparacion de 2-bencil-4-(4-piridil)-tiazoles. - Google Patents
Un procedimiento para la preparacion de 2-bencil-4-(4-piridil)-tiazoles.Info
- Publication number
- ES8700255A1 ES8700255A1 ES545439A ES545439A ES8700255A1 ES 8700255 A1 ES8700255 A1 ES 8700255A1 ES 545439 A ES545439 A ES 545439A ES 545439 A ES545439 A ES 545439A ES 8700255 A1 ES8700255 A1 ES 8700255A1
- Authority
- ES
- Spain
- Prior art keywords
- benzyl
- thiazole
- pyriol
- morpholino
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- FZWLAAWBMGSTSO-UHFFFAOYSA-N Thiazole Chemical compound C1=CSC=N1 FZWLAAWBMGSTSO-UHFFFAOYSA-N 0.000 title 1
- PZMNUBLMVHPYKL-UHFFFAOYSA-N 2-benzyl-4-pyridin-4-yl-1,3-thiazole Chemical class C=1C=CC=CC=1CC(SC=1)=NC=1C1=CC=NC=C1 PZMNUBLMVHPYKL-UHFFFAOYSA-N 0.000 abstract 1
- NAFCUKZZHZYPKB-UHFFFAOYSA-N 2-bromo-1-pyridin-4-ylethanone Chemical compound BrCC(=O)C1=CC=NC=C1 NAFCUKZZHZYPKB-UHFFFAOYSA-N 0.000 abstract 1
- 230000005494 condensation Effects 0.000 abstract 1
- 238000009833 condensation Methods 0.000 abstract 1
- AEOCXXJPGCBFJA-UHFFFAOYSA-N ethionamide Chemical compound CCC1=CC(C(N)=S)=CC=N1 AEOCXXJPGCBFJA-UHFFFAOYSA-N 0.000 abstract 1
- SUSQOBVLVYHIEX-UHFFFAOYSA-N phenylacetonitrile Chemical compound N#CCC1=CC=CC=C1 SUSQOBVLVYHIEX-UHFFFAOYSA-N 0.000 abstract 1
- 150000007979 thiazole derivatives Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/44—Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
- C07D213/46—Oxygen atoms
- C07D213/50—Ketonic radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/65—One oxygen atom attached in position 3 or 5
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Immunology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/634,094 US4697012A (en) | 1984-07-25 | 1984-07-25 | Morpholino pyridyl thiazole compound |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES545439A0 ES545439A0 (es) | 1986-10-01 |
| ES8700255A1 true ES8700255A1 (es) | 1986-10-01 |
Family
ID=24542414
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES545439A Expired ES8700255A1 (es) | 1984-07-25 | 1985-07-22 | Un procedimiento para la preparacion de 2-bencil-4-(4-piridil)-tiazoles. |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US4697012A (en]) |
| EP (1) | EP0169502B1 (en]) |
| JP (1) | JPS6137784A (en]) |
| KR (1) | KR860001105A (en]) |
| AU (1) | AU575666B2 (en]) |
| DE (1) | DE3580317D1 (en]) |
| DK (1) | DK336685A (en]) |
| ES (1) | ES8700255A1 (en]) |
| GR (1) | GR851809B (en]) |
| IL (1) | IL75823A0 (en]) |
| PT (1) | PT80833B (en]) |
| ZA (1) | ZA855581B (en]) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3486009T2 (de) * | 1983-09-09 | 1993-04-15 | Takeda Chemical Industries Ltd | 5-pyridyl-1,3-thiazol-derivate, ihre herstellung und anwendung. |
| GB9201692D0 (en) * | 1992-01-27 | 1992-03-11 | Smithkline Beecham Intercredit | Compounds |
| CN1065242C (zh) * | 1995-05-26 | 2001-05-02 | 拜尔公司 | 吡啶基－噻唑 |
| US7465736B2 (en) | 2002-06-14 | 2008-12-16 | Laboratoires Serono S.A. | Azole methylidene cyanide derivatives and their use as protein kinase modulators |
| AR045651A1 (es) * | 2003-09-19 | 2005-11-02 | Solvay Pharm Bv | Derivados de tiazol como moduladores del receptor de cannabinoide |
| US7294640B2 (en) | 2004-02-06 | 2007-11-13 | Merck & Co., Inc. | Mitotic kinesin inhibitors |
| AR083023A1 (es) * | 2010-09-17 | 2013-01-23 | Purdue Pharma Lp | Compuestos de piridina y una composicion farmaceutica que los comprende |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1112128A (en) * | 1965-12-22 | 1968-05-01 | Bellon Labor Sa Roger | New thiazolyl-diphenylmethane derivatives |
| IL28803A (en) * | 1966-11-18 | 1974-05-16 | Wyeth John & Brother Ltd | Oxazole and thiazole compounds,their preparation and pharmaceutical compositions containing them |
| CA962269A (en) * | 1971-05-05 | 1975-02-04 | Robert E. Grahame (Jr.) | Thiazoles, and their use as insecticides |
| US4153703A (en) * | 1977-06-30 | 1979-05-08 | Uniroyal, Inc. | Method of controlling insects and acarids with certain aryl-substituted thiazoles |
| DE3486009T2 (de) * | 1983-09-09 | 1993-04-15 | Takeda Chemical Industries Ltd | 5-pyridyl-1,3-thiazol-derivate, ihre herstellung und anwendung. |
-
1984
- 1984-07-25 US US06/634,094 patent/US4697012A/en not_active Expired - Fee Related
-
1985
- 1985-07-16 IL IL75823A patent/IL75823A0/xx unknown
- 1985-07-18 EP EP85108969A patent/EP0169502B1/en not_active Expired - Lifetime
- 1985-07-18 PT PT80833A patent/PT80833B/pt unknown
- 1985-07-18 DE DE8585108969T patent/DE3580317D1/de not_active Expired - Fee Related
- 1985-07-22 GR GR851809A patent/GR851809B/el unknown
- 1985-07-22 ES ES545439A patent/ES8700255A1/es not_active Expired
- 1985-07-24 AU AU45320/85A patent/AU575666B2/en not_active Expired - Fee Related
- 1985-07-24 DK DK336685A patent/DK336685A/da not_active Application Discontinuation
- 1985-07-24 ZA ZA855581A patent/ZA855581B/xx unknown
- 1985-07-24 KR KR1019850005279A patent/KR860001105A/ko not_active Ceased
- 1985-07-25 JP JP16308885A patent/JPS6137784A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| PT80833B (en) | 1987-05-27 |
| ES545439A0 (es) | 1986-10-01 |
| EP0169502B1 (en) | 1990-10-31 |
| AU575666B2 (en) | 1988-08-04 |
| PT80833A (en) | 1985-08-01 |
| US4697012A (en) | 1987-09-29 |
| IL75823A0 (en) | 1985-11-29 |
| DK336685A (da) | 1986-01-26 |
| EP0169502A2 (en) | 1986-01-29 |
| EP0169502A3 (en) | 1987-02-25 |
| ZA855581B (en) | 1986-03-26 |
| JPS6137784A (ja) | 1986-02-22 |
| DK336685D0 (da) | 1985-07-24 |
| DE3580317D1 (en) | 1990-12-13 |
| AU4532085A (en) | 1986-01-30 |
| GR851809B (en]) | 1985-11-26 |
| KR860001105A (ko) | 1986-02-22 |
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